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作者: Contreras, Jean-Marie ; Federico, Antonella ; Al-Karadaghi, Salam ; Lupino, Elisa ; Morice, Christophe ; Barge, Alessandro ; Sainas, Stefano ; Kubbutat, Michael ; Piccinini, Marco ; Pippione, Agnese C. ; Ducime, Alex ; Lolli, Marco L. ; Boschi, Donatella
Resulting from hit-to-lead optimization, the aminopyrazole3ais a NIK inhibitor selective over 44 kinases.