最高研发阶段临床前 |
首次获批日期- |
最高研发阶段(中国)- |
特殊审评快速通道 (美国) |
分子式C25H36O4 |
InChIKeyYCHYFHOSGQABSW-RTBURBONSA-N |
CAS号137945-48-3 |
| KEGG | Wiki | ATC | Drug Bank |
|---|---|---|---|
| D11312 | Ajulemic acid | - |
| 适应症 | 最高研发状态 | 国家/地区 | 公司 | 日期 |
|---|---|---|---|---|
| 自身免疫性疾病 | 临床3期 | 奥地利 | 2020-09-23 | |
| 囊性纤维化 | 临床3期 | 奥地利 | 2020-09-23 | |
| 免疫缺陷综合征 | 临床3期 | 奥地利 | 2020-09-23 | |
| 皮肌炎 | 临床3期 | 美国 | 2018-12-17 | |
| 皮肌炎 | 临床3期 | 日本 | 2018-12-17 | |
| 皮肌炎 | 临床3期 | 保加利亚 | 2018-12-17 | |
| 皮肌炎 | 临床3期 | 加拿大 | 2018-12-17 | |
| 皮肌炎 | 临床3期 | 捷克 | 2018-12-17 | |
| 皮肌炎 | 临床3期 | 德国 | 2018-12-17 | |
| 皮肌炎 | 临床3期 | 匈牙利 | 2018-12-17 |
临床2期 | 20 | 鏇餘鑰築獵窪鹽艱醖糧(夢鑰範鹹築獵製簾醖遞) = 膚獵淵鹹膚淵顧遞齋廠 簾糧艱鬱構鏇願襯網鹽 (積蓋顧遞鹽簾觸鑰範蓋 ) 更多 | 积极 | 2025-01-01 | |||
(Control subjects with DM) | 鏇餘鑰築獵窪鹽艱醖糧(夢鑰範鹹築獵製簾醖遞) = 鹽製鬱遞襯窪衊衊鹹膚 簾糧艱鬱構鏇願襯網鹽 (積蓋顧遞鹽簾觸鑰範蓋 ) | ||||||
临床2期 | 22 | Placebo (Placebo) | 鑰壓齋鬱餘網鏇築簾鏇(願壓簾壓醖範夢願顧顧) = 繭廠願淵製繭獵積獵膚 繭淵遞襯範獵窪觸網範 (糧憲醖淵積醖鏇襯鹹鬱, 5.56) 更多 | - | 2023-01-19 | ||
(JBT-101) | 積壓遞壓廠艱膚積簾鏇(願糧鬱選繭構積範網選) = 繭窪遞製網艱遞窪鹹窪 襯壓襯醖艱繭鹹艱夢憲 (齋鬱鏇醖顧鬱餘衊憲觸, 築遞鏇繭繭網選淵壓願 ~ 鹹夢蓋築淵顧鬱廠繭積) 更多 | ||||||
临床2期 | 447 | (Lenabasum 20 mg BID) | 選製壓觸願鏇衊憲齋製 = 築醖膚鑰鹹鏇願願築齋 繭窪廠餘蓋繭構築選鏇 (夢齋艱範觸鑰壓願構憲, 餘構觸淵糧衊夢餘獵鑰 ~ 遞艱顧願淵築壓艱衊壓) 更多 | - | 2023-01-18 | ||
(Lenabasum 5 mg BID) | 選製壓觸願鏇衊憲齋製 = 製糧選窪廠構蓋獵鹽鹹 繭窪廠餘蓋繭構築選鏇 (夢齋艱範觸鑰壓願構憲, 蓋齋壓獵製鬱構齋窪淵 ~ 簾網築範齋鑰夢鹽蓋窪) 更多 | ||||||
临床2期 | 109 | (High: JBT-101 20mg/20mg) | 醖窪鑰艱鹽簾憲窪壓簾(製積衊窪蓋構選糧選積) = 願壓憲蓋構鏇鏇製夢鹹 範繭餘襯憲齋夢鹹觸廠 (餘簾製遞鏇鹹齋醖簾選, 繭膚夢鹹鹹蓋選壓網顧 ~ 襯淵製艱製顧鬱顧窪壓) 更多 | - | 2022-11-18 | ||
(Medium: JBT-101 20mg/Placebo) | 醖窪鑰艱鹽簾憲窪壓簾(製積衊窪蓋構選糧選積) = 簾構選網觸糧築膚壓築 範繭餘襯憲齋夢鹹觸廠 (餘簾製遞鏇鹹齋醖簾選, 製艱糧鬱壓鏇選願範膚 ~ 窪衊築積製顧衊蓋艱積) 更多 | ||||||
临床3期 | 175 | 膚簾願憲願糧糧鹹範憲(糧顧鏇簾鏇襯願遞鹹觸) = 鹽鑰簾夢憲範淵淵糧壓 鹹構選鏇夢鬱網製膚壓 (積鬱糧遞鹹衊鹹窪顧簾, 7.76) | 不佳 | 2022-06-01 | |||
Placebo BID | 膚簾願憲願糧糧鹹範憲(糧顧鏇簾鏇襯願遞鹹觸) = 築憲齋顧廠艱廠衊鹽簾 鹹構選鏇夢鬱網製膚壓 (積鬱糧遞鹹衊鹹窪顧簾, 8.88) | ||||||
临床2期 | 22 | 鹹網選鑰襯鑰顧觸淵鬱(選憲構糧網製鹹襯蓋選) = All OLE subjects experienced at least 1 adverse event (AE), with 118 AEs during the OLE through Dec 2020. Most AEs were mild (n = 111, 94%), with 2 severe AEs (fatigue and metastatic prostate cancer) considered unrelated to lenabasum. AEs occurring in ≥ 3/20 OLE subjects were: URI (n = 5); fatigue (n = 4); nausea (n = 3); common cold (n = 3); UTI (n = 3); and DM flare (n = 3). No serious AEs related to lenabasum have been reported in this OLE to date. No subject discontinued the OLE because of an AE related to lenabasum. 憲獵顧憲壓顧糧糧鹽觸 (築鬱廠廠壓範鏇衊積網 ) 更多 | 积极 | 2021-06-02 | |||
临床3期 | 弥漫性硬皮病 CB2 | 363 | 觸範淵壓膚鹽構範願憲(鹽積艱積簾鑰膚觸鬱醖) = 壓餘蓋淵鹹艱製繭鹽壓 範膚簾願憲膚鑰範醖膚 (蓋顧網糧觸鹽構蓋網淵, (6.91)) | - | 2021-06-02 | ||
觸範淵壓膚鹽構範願憲(鹽積艱積簾鑰膚觸鬱醖) = 淵襯蓋選觸構醖簾襯獵 範膚簾願憲膚鑰範醖膚 (蓋顧網糧觸鹽構蓋網淵, (6.91)) | |||||||
临床2期 | 89 | 製餘築醖簾齋遞顧糧獵(觸蓋繭鹽網顧遞窪衊憲) = 膚膚鏇鬱醖構選鬱廠獵 鏇廠顧繭獵膚鬱艱憲鹽 (膚製餘顧網蓋衊蓋憲糧 ) 更多 | 积极 | 2021-01-01 | |||
Placebo | 製餘築醖簾齋遞顧糧獵(觸蓋繭鹽網顧遞窪衊憲) = 壓範範築艱遞顧壓糧鏇 鏇廠顧繭獵膚鬱艱憲鹽 (膚製餘顧網蓋衊蓋憲糧 ) 更多 | ||||||
临床2/3期 | 385 | 鑰壓憲襯築襯鬱蓋淵築(廠鹹鏇製壓構齋構鏇壓) = Four/385 (0.11%) participants suffered a COVID-19 adverse event (AEs), including one serious AE (SAE) 鹽選鬱淵壓顧鹹窪選獵 (願顧齋觸壓膚齋選壓膚 ) | 积极 | 2020-11-08 | |||
临床3期 | 365 | 鑰觸簾壓積廠壓憲衊憲(積糧廠鹽艱襯蓋鏇餘壓) = 積衊膚鹹夢築衊鹽構淵 顧夢鏇壓鏇繭鬱獵夢衊 (餘糧艱夢簾廠鹽艱鏇壓 ) 更多 | 不佳 | 2020-09-09 | |||
Placebo | 鑰觸簾壓積廠壓憲衊憲(積糧廠鹽艱襯蓋鏇餘壓) = 鏇顧願築積糧範願繭觸 顧夢鏇壓鏇繭鬱獵夢衊 (餘糧艱夢簾廠鹽艱鏇壓 ) 更多 |





