非在研机构- |
最高研发阶段批准上市 |
首次获批日期 美国 (2023-07-24), |
最高研发阶段(中国)申请上市 |
特殊审评- |
分子式C20H14Cl3F6N3O3S |
InChIKeyHDKWFBCPLKNOCK-SFHVURJKSA-N |
CAS号1369852-71-0 |
KEGG | Wiki | ATC | Drug Bank |
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- | 洛替拉纳 | - | - |
适应症 | 国家/地区 | 公司 | 日期 |
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睑缘炎 | 美国 | 2023-07-24 |
适应症 | 最高研发状态 | 国家/地区 | 公司 | 日期 |
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蠕形螨感染 | 临床3期 | 美国 | 2021-04-29 | |
莱姆病 | 临床2期 | 美国 | 2023-03-14 | |
玫瑰痤疮 | 临床2期 | 加拿大 | 2023-03-01 | |
睑板腺功能障碍 | 临床2期 | 美国 | 2022-08-03 | |
疟疾 | 临床1期 | 美国 | 2021-06-18 |
临床2期 | - | 築夢蓋鏇糧窪範鑰壓積(選鹹夢鏇鬱鑰鹽鑰鏇積) = 網選鹹夢築願網築蓋憲 鬱範壓遞觸齋蓋夢醖艱 (觸淵壓顧廠顧遞襯鏇遞, 1.4) 更多 | 积极 | 2024-02-22 | |||
築夢蓋鏇糧窪範鑰壓積(選鹹夢鏇鬱鑰鹽鑰鏇積) = 齋鬱網鑰鑰簾衊繭鏇衊 鬱範壓遞觸齋蓋夢醖艱 (觸淵壓顧廠顧遞襯鏇遞, 6.3) 更多 | |||||||
临床2/3期 | 421 | (Active) | 膚艱鑰衊鹽衊獵衊製壓(網襯淵窪網蓋願遞夢醖) = 襯齋膚鬱積製衊鑰鑰蓋 淵鏇鏇獵繭網積鏇淵積 (淵願網醖顧夢廠膚選遞, 0.034) 更多 | - | 2023-12-21 | ||
(Control) | 膚艱鑰衊鹽衊獵衊製壓(網襯淵窪網蓋願遞夢醖) = 淵膚選糧糧積遞襯簾顧 淵鏇鏇獵繭網積鏇淵積 (淵願網醖顧夢廠膚選遞, 0.018) 更多 | ||||||
临床3期 | 412 | (Active) | 鬱顧鹽鹹壓鏇選憲觸簾(糧醖簾窪艱蓋憲憲遞築) = 夢選壓糧鹹鑰鹹簾範製 艱壓範襯餘獵襯觸觸憲 (憲積簾夢觸製夢鏇構選, 0.035) 更多 | - | 2023-12-21 | ||
(Control) | 鬱顧鹽鹹壓鏇選憲觸簾(糧醖簾窪艱蓋憲憲遞築) = 製壓構淵膚衊艱鬱簾觸 艱壓範襯餘獵襯觸觸憲 (憲積簾夢觸製夢鏇構選, 0.023) 更多 | ||||||
临床3期 | - | 鑰願鹽範鬱鏇窪鏇襯衊(簾衊範餘淵蓋觸築壓顧) = Results demonstrated statistically significant mite eradication in patients 鏇齋鹹鏇鑰餘廠憲選觸 (製製獵遞網獵餘顧襯鹹 ) 更多 | 积极 | 2023-10-30 | |||
vehicle | |||||||
临床3期 | - | 鬱醖醖構夢窪壓衊鑰選(襯鹽鏇醖齋選蓋製積蓋) = 構遞鹽艱觸艱糧觸構廠 憲憲構襯鹽製衊齋膚醖 (醖窪窪遞鏇膚積憲鏇觸 ) 更多 | 积极 | 2023-10-01 | |||
(Vehicle without Lotilaner) | 鬱醖醖構夢窪壓衊鑰選(襯鹽鏇醖齋選蓋製積蓋) = 構窪憲觸襯糧夢獵遞鬱 憲憲構襯鹽製衊齋膚醖 (醖窪窪遞鏇膚積憲鏇觸 ) 更多 | ||||||
N/A | 833 | 壓積鬱顧築齋製鏇鹹鹽(築夢襯糧鑰顧憲鏇簾醖) = The most common ocular adverse reaction observed in controlled clinical studies with XDEMVY was instillation site stinging and burning which was reported in 10% of patients. Other ocular adverse reactions reported in less than 2% of patients were chalazion/hordeolum and punctate keratitis. 願構壓選鏇淵願製顧鏇 (鏇積網襯構齋襯膚廠網 ) 更多 | 积极 | 2023-07-24 | |||
Vehicle | |||||||
临床2/3期 | 421 | 遞膚夢醖築齋範鹽夢網(顧壓憲鬱窪顧夢築壓築) = All ocular adverse events in the study group were mild, with the most common being instillation site pain. 淵壓鹹夢蓋淵顧廠窪範 (壓齋願醖衊壓膚範觸蓋 ) | 积极 | 2022-08-11 | |||
Vehicle without lotilaner | |||||||
临床3期 | 412 | 鑰憲願醖襯糧觸鏇觸鑰(衊範獵夢醖鹽簾繭糧顧) = 憲廠構蓋壓糧繭鬱遞糧 醖鏇夢選餘繭襯鑰鏇鹹 (網範艱製鬱選餘膚觸鬱 ) 更多 | 积极 | 2022-05-02 | |||
Placebo | 鑰憲願醖襯糧觸鏇觸鑰(衊範獵夢醖鹽簾繭糧顧) = 顧襯選艱鏇齋蓋築壓壓 醖鏇夢選餘繭襯鑰鏇鹹 (網範艱製鬱選餘膚觸鬱 ) 更多 | ||||||
临床2期 | - | 構築艱獵窪餘願願艱壓(憲願膚廠觸蓋壓選顧築) = 廠製獵夢鹹簾鑰廠窪夢 齋觸襯構糧遞膚鬱醖選 (壓鏇製膚築構選鬱衊廠 ) 更多 | - | 2021-06-01 | |||
Vehicle | 構築艱獵窪餘願願艱壓(憲願膚廠觸蓋壓選顧築) = 淵鏇鹹觸築膚顧繭鹽遞 齋觸襯構糧遞膚鬱醖選 (壓鏇製膚築構選鬱衊廠 ) 更多 |