别名 G protein-coupled receptor 39、G-protein coupled receptor 39、GPR39 |
简介 Zn(2+) acts as an agonist. This receptor mediates its action by association with G proteins that activate a phosphatidylinositol-calcium second messenger system. Its effect is mediated mainly through G(q)-alpha and G(12)/G(13) proteins. Involved in regulation of body weight, gastrointestinal mobility, hormone secretion and cell death (By similarity). |
靶点- |
作用机制 GPR39 激动剂 |
在研机构 Cerevance, Inc.初创企业 |
原研机构 Cerevance, Inc.初创企业 |
在研适应症 |
非在研适应症- |
最高研发阶段临床前 |
首次获批国家/地区- |
首次获批日期1800-01-20 |