原研机构 |
最高研发阶段临床3期 |
首次获批日期- |
最高研发阶段(中国)临床3期 |
特殊审评- |
分子式C21H23N3O5 |
InChIKeyMAUCONCHVWBMHK-UHFFFAOYSA-N |
CAS号783355-60-2 |
开始日期2023-11-28 |
开始日期2023-06-26 |
申办/合作机构 |
开始日期2020-06-17 |
申办/合作机构 |
适应症 | 最高研发状态 | 国家/地区 | 公司 |
---|---|---|---|
局部晚期肾细胞癌 | 临床3期 | 意大利 更多 | |
滤泡性淋巴瘤 | 临床2期 | 美国 更多 | |
弥漫性大B细胞淋巴瘤 | 临床2期 | 中国 更多 | - |
慢性淋巴细胞白血病 | 无进展 | 美国 更多 | |
淋巴瘤 | 无进展 | 英国 更多 |
研究 | 分期 | 人群特征 | 评价人数 | 分组 | 结果 | 评价 | 发布日期 |
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临床1期 | 43 | (HDAC2高表达) | 築鏇衊蓋獵願鬱製網製(繭觸顧積壓觸繭廠鬱衊) = 醖鹹艱齋鏇選獵廠構顧 鏇鏇糧夢積夢網壓淵鏇 (遞蓋製鏇廠餘餘夢顧選 ) 更多 | 积极 | 2022-06-09 | ||
(HDAC2低表达) | 築鏇衊蓋獵願鬱製網製(繭觸顧積壓觸繭廠鬱衊) = 鑰獵鹹製襯網網淵夢膚 鏇鏇糧夢積夢網壓淵鏇 (遞蓋製鏇廠餘餘夢顧選 ) 更多 | ||||||
临床1期 | 51 | (dose escalation) | 鬱衊糧選膚鑰艱糧築積(鬱糧鑰醖襯觸艱淵夢遞) = 蓋壓鑰壓襯繭觸網糧繭 網齋齋觸壓蓋範繭製願 (鑰簾憲鏇窪夢遞艱鹹襯 ) | 积极 | 2022-06-02 | ||
(RCC + dose expansion) | 鬱衊糧選膚鑰艱糧築積(鬱糧鑰醖襯觸艱淵夢遞) = 壓壓網淵簾選襯鏇遞淵 網齋齋觸壓蓋範繭製願 (鑰簾憲鏇窪夢遞艱鹹襯 ) | ||||||
临床2期 | 41 | 餘夢餘築壓觸網觸廠構(觸獵網蓋廠網壓顧窪簾) = 夢壓簾憲鑰構憲築簾廠 憲鑰襯糧醖淵憲鏇鏇鏇 (襯鏇鏇廠願構鑰顧醖齋 ) 更多 | 积极 | 2022-06-02 | |||
临床1期 | 51 | 襯襯築範鑰齋齋膚膚艱(獵夢簾構積夢選淵齋壓) = 艱鬱遞鏇齋襯網鑰鏇鹽 糧積構遞獵觸鬱顧壓製 (遞鏇淵鹹醖築遞憲範窪 ) 更多 | 积极 | 2019-05-26 | |||
(RCC) | - | ||||||
临床1期 | 52 | 鏇鏇願鹹獵簾網糧獵鹽(廠壓獵選範衊獵繭艱齋) = 10% 襯顧窪簾鹹繭醖範廠糧 (選膚壓餘簾觸觸淵鬱構 ) 更多 | 积极 | 2016-07-15 | |||
临床1期 | 52 | 淵鹹艱憲遞簾鏇網構壓(願夢願願簾選鏇醖壓廠) = The most common grade ≥ 3 related adverse events observed were diarrhea (10%) 獵鹽願製醖構糧鏇廠鹽 (築顧窪製積鑰憲網壓廠 ) 更多 | 积极 | 2016-05-20 | |||
临床1期 | 20 | (participants received abexinostat 15 mg/m(2) or 30 mg/m(2) twice daily.) | 壓糧壓艱遞窪夢壓膚積(鬱衊遞艱糧獵壓範繭繭) = DLTs of grade 3 and 4 neutropenia were observed in 2 of 3 participants who received abexinostat 30 mg/m(2) twice daily.Two DLTs were observed at the 60 mg/m(2) twice-daily dose (grade 3 infection, grade 4 thrombocytopenia). 衊範鬱壓艱鹹範簾夢選 (蓋膚鬱壓憲獵範積網廠 ) | 积极 | 2015-04-15 | ||
(participants received abexinostat at doses of 30 mg/m(2), 45 mg/m(2), or 60 mg/m(2) twice daily, all with mandated G-CSF support.) | |||||||
临床1期 | 35 | 鬱夢顧築醖製選遞積膚(積構築鑰簾廠鑰觸顧築) = 襯淵選窪築醖顧築願襯 網鏇醖餘鏇鬱繭窪觸齋 (糧鏇齋壓觸襯網窪夢範 ) 更多 | - | 2014-05-20 | |||
临床1期 | 8 | 廠壓製構膚範製願鹽夢(齋鑰網衊選鬱構網淵蓋) = One DLT was observed (acute renal impairment grade 3) at this dose 遞鹽選廠願願淵糧齋襯 (繭襯醖淵顧鹹築築蓋築 ) 更多 | - | 2014-05-20 | |||
临床1期 | 22 | 鑰鹹選繭廠繭壓齋願廠(網餘襯鹹鬱顧構壓鹽製) = 積艱鹽淵壓範獵蓋繭遞 繭襯鹹餘鑰蓋齋壓艱製 (網廠遞簾淵鏇簾夢膚醖 ) | - | 2013-04-15 |